Metabolic / GLP-1
Retatrutide
A triple agonist of GIP, GLP-1, and glucagon receptors currently in late-phase research for obesity and metabolic indications.
Quick facts
Molecular weight
4,731 Da
Half-life
144 h
Frequency
weekly
Admins / wk
1
Routes
SubQ
Typical dose
500 mcg–12.0 mg
Mechanism & positioning
A triple agonist of GIP, GLP-1, and glucagon receptors currently in late-phase research for obesity and metabolic indications.
Researched for: triple GIP/GLP-1/glucagon agonism, adipose mobilisation.
Reconstitution defaults
Default vial
10 mg
BAC water
2 mL
Concentration
5000 mcg/mL
Doses per vial
~20
Other stocked vial sizes: 24, 40, 60 mg.
Calculate with this peptide
Dosage Calculator
Pre-filled for 500 mcg from a 10 mg vial in 2 mL BAC water.
Reconstitution Calculator
Auto-fills 10 mg + 2 mL BAC water + 500 mcg target dose.
Half-Life Calculator
Simulates steady-state at 500 mcg weekly.
Titration Schedule Builder
Stepwise escalation from 500 mcg to 12.0 mg.
Pen & Cartridge Calculator
Loads the Retatrutide 24 mg pen preset (24 mg / 3 mL).
Documented pairwise interactions
- avoid
Retatrutide + Semaglutide
Overlapping GLP-1 receptor agonism; combined effects unpredictable in current literature.
- avoid
Retatrutide + Tirzepatide
Both are multi-receptor incretin agonists; concurrent use exceeds any published research protocol.
References
- Jastreboff AM et al., NEJM, 2023.
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